Archiv der Pharmazie
@arch_pharm
International journal focusing on all fields of pharmaceutical and medicinal chemistry. Published by @WileyVCH with the DPhG.
ID: 1422096239408074757
https://onlinelibrary.wiley.com/journal/15214184 02-08-2021 07:27:15
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A colorful season is coming up 🍂🍁When chlorophyll is degraded in autumn, #phyllobilin levels rise! Curious to know more? A review in Archiv der Pharmazie by @PhylloLab gives an extensive overview of current knowledge on structures, occurrence, and #bioactivities. onlinelibrary.wiley.com/doi/10.1002/ar…
Thorough 2D NMR characterization of 1-oxo-1H-phenalene derivatives led to structure corrections and nanomolar inhibitors of BCL-2. Study and guidelines for proper structure determination in Archiv der Pharmazie were conducted by Izidor Sosič Christian Steinebach Rheinische Friedrich-Wilhelms-Universität Bonn. onlinelibrary.wiley.com/doi/10.1002/ar…
Another big #GPCR meeting 🤩 Looking forward to present our data from Schulte lab on using conformational receptor biosensors to study #Frizzled activation & signalling!
The Bracher group Universität München identified, by means of chemical synthesis and crystal structure analysis, the active stereoisomer of the TRPML1 inhibitor ML-SI3. This small molecule is an important tool to modulate this potential drug target Archiv der Pharmazie. onlinelibrary.wiley.com/doi/10.1002/ar…
Laura Schäkel et al. from agmueller.unibonn Rheinische Friedrich-Wilhelms-Universität Bonn have recently published 2-substituted thienotetrahydropyridine derivatives as allosteric ectonucleotidase inhibitors with improved selectivity profile in Archiv der Pharmazie. onlinelibrary.wiley.com/doi/10.1002/ar…
The "Archiv der Pharmazie" Archiv der Pharmazie is turning 200 and we want to celebrate it with you. Below is the link to the invitation to our GPCR Special Collection served by Steffen Pockes as a guest editor. There is no submission deadline. Wiley Chemistry onlinelibrary.wiley.com/doi/toc/10.100…
Flashback: Archiv der Pharmazie ahead of Angewandte Chemie on paullones: In 1992 the first report on the synthesis of indolo[3,2-d][1]benzazepines (dubbed paullones) by C. Kunick appeared shortly before the same heterocyclic system was reported by A. P. Kozikowski. #AdP200 Wiley Chemistry
Jürg Zimmermann's 1996 report on selective kinase inhibitors in Archiv der Pharmazie is cited in Nature Reviews Drug Discovery to have paved the way to identify and optimize synthetic small-molecule kinase inhibitors like imatinib. #AdP200 Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…
The Wünsch lab has combined pharmacophores of two potent NMDA receptor antagonists to design oxazolobenzazepines Archiv der Pharmazie. These negative allosteric modulators of GluN2B-NMDA receptors may be useful in neurodegenerative disorders. Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…
Congratulations to the #FiMC2022 Innovation Prize winners, Dr. Steffen Pockes Steffen Pockes and Dr. Oliver Thorn-Seshold Thorn-Seshold Lab 🇺🇦! #medchem #chembio #pharma #drugdiscovery #medchemtalents #euromedchemtalents EFMC Young Scientists Network EFMC
The Wende lab has published physical cold plasma for controllable prodrug activation in Archiv der Pharmazie: First exploratory example for a prodrug release triggered by tissue-compatible cold plasma in vitro. Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…
Working together with my alma mater group 👩🏻🔬 from @UNSbahiablanca. Interesting first multidisciplinary approach for TADDOL derivatives. Archiv der Pharmazie Andrea Costantino nitin charbe Yorley Duarte @prasher_sharma Mandolesi Sandra Kamal Dua Facultad de Química y de Farmacia UC IIBM UC Universidad de Talca CBIB UNAB Universidad Católica
A new class of 1,4-Dihydropyridinebutyrolactone-derived ring-opened ester and amide analogs from the Georg lab Gunda I. Georg to target BET bromodomains were just recently published in Archiv der Pharmazie. University of Minnesota Medicinal Chemistry Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…
We are looking forward to the upcoming DPhG conference in Marburg Philipps-Universität. And right at the beginning tomorrow, Tuesday, our editor-in-chief Andreas Link sums up the role of our journal Archiv der Pharmazie in the 21st century. Come in large numbers! Wiley Chemistry
Preventing brain damage and dysfunction after traumatic brain injury using potassium channel openers could become clinical practice if nontoxic analogs of retigabine could be found. Wurm et al. shed some light on the way to go.Archiv der Pharmazie Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…
The Koch lab Universität Münster is introducing to artificial intelligence and deep learning using interactive electronic programming notebooks in Archiv der Pharmazie. Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…
The Georg lab Gunda I. Georg is reporting selective retinoic acid receptor alpha antagonist ER-50891 and related analogs for male contraception. University of Minnesota Medicinal Chemistry Archiv der Pharmazie Wiley Chemistry onlinelibrary.wiley.com/doi/10.1002/ar…